TAPI-1 trifluoroacetate (163847-77-6(free base))
Code | Size | Price |
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TAR-T4122-1mg | 1mg | £189.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4122-2mg | 2mg | £285.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T4122-5mg | 5mg | £546.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
TAPI-1 is an ADAM17/TACE inhibitor, which blocks shedding of cytokine receptors.
CAS:
T4122
Formula:
C28H38F3N5O7
Molecular Weight:
613.62
Pathway:
Proteases/Proteasome
Purity:
0.9806
SMILES:
OC(=O)C(F)(F)F.CC(C)CC(CC(=O)NO)C(=O)N[C@@H](Cc1ccc2ccccc2c1)C(=O)N[C@@H](C)C(=O)NCCN
Target:
MMP
References
M?llberg J, et al. J Immunol. 1995, 155(11), 5198-5205
Oikawa H, et al. Life Sci. 2014, 97(2), 137-144.
Slack BE, et al. Biochem J. 2001, 357(Pt 3), 787-794.