hnps-PLA Inhibitor

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TargetMol
Product Code: TAR-T4192
Supplier: TargetMol
CodeSizePrice
TAR-T4192-1mg1mg£111.00
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TAR-T4192-2mg2mg£130.00
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TAR-T4192-5mg5mg£168.00
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TAR-T4192-1mL1 mL * 10 mM (in DMSO)£182.00
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TAR-T4192-10mg10mg£242.00
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TAR-T4192-25mg25mg£359.00
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TAR-T4192-50mg50mg£500.00
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TAR-T4192-100mg100mg£683.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Hnps-PLA Inhibitor is an inhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
CAS:
185298-58-2
Formula:
C21H21N3O4
Molecular Weight:
379.416
Pathway:
Metabolism; Immunology/Inflammation
Purity:
0.9895
SMILES:
CCc1c(C(=O)C(N)=O)c2c(OCC(N)=O)cccc2n1Cc1ccccc1
Target:
Phospholipase; LTR

References

Mihelich ED, et al. Structure-based design of a new class of anti-inflammatory drugs: secretory phospholipase A(2) inhibitors, SPI. Biochim Biophys Acta. 1999 Nov 23;1441(2-3):223-8 Meng H, Liu Y, Zhai Y, Lai L. Optimization of 5-hydroxytryptamines as dual function inhibitors targeting phospholipase A2 and leukotriene A4 hydrolase. Eur J Med Chem. 2013 Jan;59:160-7