Protein kinase inhibitors 1
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TAR-T4636-100mg | 100mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
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TAR-T4636-50mg | 50mg | Enquire | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
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Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Protein kinase inhibitors 1 is a novel inhibitor of HIPK2 with an IC50 of 74 nM and Kd of 9.5 nM.
CAS:
1365986-44-2
Formula:
C18H17N5O3S
Molecular Weight:
383.43
Pathway:
; Tyrosine Kinase/Adaptors; Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
O=C1NC(=O)C(S1)=Cc1c[nH]c(=O)c(c1)-c1ccc(nc1)N1CCNCC1
Target:
DYRK
References
Miduturu CV, et al. High-throughput kinase profiling: a more efficient approach toward the discovery of new kinaseinhibitors. Chem Biol. 2011 Jul 29;18(7):868-79.