GSK467

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TargetMol
Product Code: TAR-T5484
Supplier: TargetMol
CodeSizePrice
TAR-T5484-1mg1mg£130.00
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TAR-T5484-5mg5mg£213.00
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TAR-T5484-1mL1 mL * 10 mM (in DMSO)£229.00
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TAR-T5484-10mg10mg£282.00
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TAR-T5484-25mg25mg£495.00
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TAR-T5484-50mg50mg£686.00
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TAR-T5484-100mg100mg£930.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GSK467 is a potent and selective inhibitor of KDM5 (JARID1)(Ki : 10 nM).
CAS:
1628332-52-4
Formula:
C17H13N5O2
Molecular Weight:
319.324
Pathway:
Chromatin/Epigenetic
Purity:
1
SMILES:
O=c1[nH]c(Oc2cnn(Cc3ccccc3)c2)nc2cnccc12
Target:
Histone Demethylase; Histone Methyltransferase

References

Johansson C, et al. Structural analysis of human KDM5B guides histone demethylase inhibitor development. Nat Chem Biol. 2016 Jul;12(7):539-45.