CGP71683 hydrochloride

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TargetMol
Product Code: TAR-T5587
Supplier: TargetMol
CodeSizePrice
TAR-T5587-1mg1mg£109.00
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TAR-T5587-2mg2mg£125.00
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TAR-T5587-5mg5mg£156.00
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TAR-T5587-1mL1 mL * 10 mM (in DMSO)£166.00
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TAR-T5587-10mg10mg£201.00
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TAR-T5587-25mg25mg£287.00
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TAR-T5587-50mg50mg£386.00
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TAR-T5587-100mg100mg£551.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
CGP71683 is a competitive neuropeptide Y5 receptor antagonist (Ki: 1.3 nM) and shows no obvious activity at Y1 receptor (Ki >4000 nM) and Y2 receptor (Ki: 200 nM) in cell membranes.
CAS:
192322-50-2
Formula:
C26H30ClN5O2S
Molecular Weight:
512.07
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9982
SMILES:
Cl.Nc1nc(NC[C@H]2CC[C@H](CNS(=O)(=O)c3cccc4ccccc34)CC2)nc2ccccc12
Target:
Neuropeptide Y Receptor

References

Kask A, et al. Neuropeptide Y Y(5) receptor antagonist CGP71683A: the effects on food intake and anxiety-related behavior in the rat. Eur J Pharmacol. 2001 Mar 2;414(2-3):215-24. Lecklin A, et al. Receptor subtypes Y1 and Y5 mediate neuropeptide Y induced feeding in the guinea-pig. Br J Pharmacol. 2002 Apr;135(8):2029-37.