PD318088

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TargetMol
Product Code: TAR-T6152
Supplier: TargetMol
CodeSizePrice
TAR-T6152-1mg1mg£107.00
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TAR-T6152-2mg2mg£137.00
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TAR-T6152-5mg5mg£177.00
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TAR-T6152-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T6152-10mg10mg£273.00
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TAR-T6152-25mg25mg£450.00
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TAR-T6152-50mg50mg£629.00
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TAR-T6152-100mg100mg£863.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
PD318088 is a non-ATP competitive allosteric MEK1/2 inhibitor, binding simultaneously with ATP in a region of the MEK1 active site that is adjacent to the ATP-binding site.
CAS:
391210-00-7
Formula:
C16H13BrF3IN2O4
Molecular Weight:
561.094
Pathway:
MAPK
Purity:
0.9969
SMILES:
OCC(O)CONC(=O)c1cc(Br)c(F)c(F)c1Nc1ccc(I)cc1F
Target:
MEK

References

Ohren JF, et al. Nat Struct Mol Biol, 2004, 11(12), 1192-1197.