CTEP

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TargetMol
Product Code: TAR-T6457
Supplier: TargetMol
CodeSizePrice
TAR-T6457-1mg1mg£99.00
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TAR-T6457-2mg2mg£112.00
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TAR-T6457-5mg5mg£136.00
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TAR-T6457-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T6457-10mg10mg£185.00
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TAR-T6457-25mg25mg£270.00
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Quantity:
TAR-T6457-50mg50mg£432.00
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TAR-T6457-100mg100mg£562.00
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TAR-T6457-500mg500mg£1,131.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CTEP (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold selectivity over other mGlu receptors.
CAS:
871362-31-1
Formula:
C19H13ClF3N3O
Molecular Weight:
391.78
Pathway:
Neuroscience
Purity:
1
SMILES:
Cc1nc(C#Cc2ccnc(Cl)c2)c(C)n1-c1ccc(OC(F)(F)F)cc1
Target:
GluR

References

Lindemann L, et al. J Pharmacol Exp Ther, 2011, 339(2), 474-486. Michalon A, et al. Neuron, 2012, 74(1), 49-56.