EI1

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TargetMol
Product Code: TAR-T6484
Supplier: TargetMol
CodeSizePrice
TAR-T6484-1mg1mg£99.00
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TAR-T6484-2mg2mg£112.00
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TAR-T6484-1mL1 mL * 10 mM (in DMSO)£127.00
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TAR-T6484-5mg5mg£136.00
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TAR-T6484-10mg10mg£177.00
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TAR-T6484-25mg25mg£267.00
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TAR-T6484-50mg50mg£386.00
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TAR-T6484-100mg100mg£526.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
EI1 is a potent and selective EZH2 inhibitor with IC50 of 15 nM and 13 nM for EZH2 (WT) and EZH2 (Y641F), respectively.
CAS:
1418308-27-6
Formula:
C23H26N4O2
Molecular Weight:
390.487
Pathway:
Apoptosis; Chromatin/Epigenetic
Purity:
0.9998
SMILES:
CCC(CC)n1ccc2c(cc(cc12)C#N)C(=O)NCc1c(C)cc(C)[nH]c1=O
Target:
Apoptosis; Histone Methyltransferase

References

Qi W, et al. Proc Natl Acad Sci U S A. 2012, 109(52), 21360-21365.