Bitopertin

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TargetMol
Product Code: TAR-T6788
Supplier: TargetMol
CodeSizePrice
TAR-T6788-1mg1mg£96.00
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TAR-T6788-2mg2mg£107.00
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TAR-T6788-5mg5mg£128.00
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TAR-T6788-1mL1 mL * 10 mM (in DMSO)£142.00
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TAR-T6788-10mg10mg£149.00
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TAR-T6788-25mg25mg£251.00
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TAR-T6788-50mg50mg£402.00
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TAR-T6788-100mg100mg£564.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Bitopertin (RG1678, RO-4917838) is a potent inhibitor of glycine transporter 1 (GlyT1), with Ki of 8.1 nM for human hGlyT1b and IC50 of 22-25 nM in Chinese hamster ovary cells.
CAS:
845614-11-1
Formula:
C21H20F7N3O4S
Molecular Weight:
543.46
Pathway:
Neuroscience
Purity:
0.9997
SMILES:
C[C@H](Oc1ccc(cc1C(=O)N1CCN(CC1)c1ncc(cc1F)C(F)(F)F)S(C)(=O)=O)C(F)(F)F
Target:
GlyT

References

Alberati D, et al. Neuropharmacology. 2012, 62(2):1152-1161. Bugarski-Kirola D, et al. Eur Neuropsychopharmacol. 2014, 24(7):1024-1036.