CPI-169 racemate

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TargetMol
Product Code: TAR-T6809
Supplier: TargetMol
CodeSizePrice
TAR-T6809-1mg1mg£111.00
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TAR-T6809-2mg2mg£128.00
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TAR-T6809-5mg5mg£173.00
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TAR-T6809-1mL1 mL * 10 mM (in DMSO)£189.00
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TAR-T6809-10mg10mg£215.00
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TAR-T6809-25mg25mg£389.00
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TAR-T6809-50mg50mg£544.00
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TAR-T6809-100mg100mg£744.00
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.
CAS:
1450655-76-1
Formula:
C27H36N4O5S
Molecular Weight:
528.67
Pathway:
Chromatin/Epigenetic
Purity:
0.9914
SMILES:
CCS(=O)(=O)N1CCC(CC1)C(C)n1c(C)c(C(=O)NCc2c(OC)cc(C)[nH]c2=O)c2ccccc12
Target:
Epigenetic Reader Domain; Histone Methyltransferase

References

Bradley WD, et al. Chem Biol. 2014, 21(11), 1463-1475.