Vorapaxar

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TargetMol
Product Code: TAR-T7013
Supplier: TargetMol
CodeSizePrice
TAR-T7013-1mg1mg£127.00
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TAR-T7013-5mg5mg£189.00
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TAR-T7013-1mL1 mL * 10 mM (in DMSO)£201.00
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TAR-T7013-10mg10mg£254.00
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TAR-T7013-25mg25mg£402.00
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TAR-T7013-50mg50mg£567.00
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TAR-T7013-100mg100mg£777.00
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TAR-T7013-500mg500mg£1,476.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Vorapaxar (SCH 530348) is an effective and orally active thrombin receptor (PAR-1) antagonist (Ki: 8.1 nM).
CAS:
618385-01-6
Formula:
C29H33FN2O4
Molecular Weight:
492.591
Pathway:
GPCR/G Protein
Purity:
0.9993
SMILES:
CCOC(=O)N[C@@H]1CC[C@@H]2[C@H](C[C@@H]3[C@@H]([C@@H](C)OC3=O)[C@H]2C=Cc2ccc(cn2)-c2cccc(F)c2)C1
Target:
Protease-activated Receptor

References

Tang W, Huang B, Wang J, et al. A label-free screening approach targeted protease-activated receptor 1 based on dynamic mass redistribution in living cells[J]. RSC Advances. 2017, 7(68): 43005-43013. Chackalamannil S, et al. J Med Chem, 2008, 51(11), 3061-3064. Tang W, Huang B, Wang J, et al. A label-free screening approach targeted protease-activated receptor 1 based on dynamic mass redistribution in living cells. RSC Advances. 2017, 7(68): 43005-43013