Imidazenil
Code | Size | Price |
---|
TAR-T8971-1mg | 1mg | £152.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8971-5mg | 5mg | £246.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8971-1mL | 1 mL * 10 mM (in DMSO) | £282.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8971-10mg | 10mg | £360.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8971-25mg | 25mg | £548.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T8971-50mg | 50mg | £766.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Imidazenil is an modulator of GABA-A that blocks the sedative effects without lowering the convulsion threshold.
CAS:
151271-08-8
Formula:
C18H12BrFN4O
Molecular Weight:
399.223
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.984
SMILES:
NC(=O)c1ncn-2c1CN=C(c1ccccc1Br)c1cc(F)ccc-21
Target:
GABA Receptor
References
Giusti P , Duci I , Puia G , et al. Imidazenil: a new partial positive allosteric modulator of gamma-aminobutyric acid (GABA) action at GABAA receptors.[J]. Journal of Pharmacology & Experimental Therapeutics, 1993, 266(2):1018-1028.
Auta J , Giusti P , Guidotti A , et al. Imidazenil, a partial positive allosteric modulator of GABAA receptors, exhibits low tolerance and dependence liabilities in the rat.[J]. Journal of Pharmacology & Experimental Therapeutics, 1994, 270(3):1262-9.