Desketoraloxifene
Code | Size | Price |
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TAR-T9001-5mg | 5mg | £313.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T9001-10mg | 10mg | £435.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T9001-25mg | 25mg | £728.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Desketoraloxifene is a selective estrogen receptor modulator, inhibiting mammalian PLD (PLD1 and PLD2).
CAS:
216570-81-9
Formula:
C27H27NO3S
Molecular Weight:
445.57
Pathway:
Metabolism
Purity:
0.98
SMILES:
C1CCN(CC1)CCOC2=CC=C(C=C2)C3=C(SC4=C3C=CC(=C4)O)C5=CC=C(C=C5)O
Target:
Phospholipase
References
Scott S A , Spencer C T , MC O?Reilly, et al. Discovery of Desketoraloxifene Analogues as Inhibitorsof Mammalian, Pseudomonas aeruginosa, and NAPE PhospholipaseD Enzymes[J]. Acs Chemical Biology, 2015, 10(2):421.
Cho C H , Jung D I , Neuenswander B , et al. Parallel synthesis of a desketoraloxifene analogue library via iodocyclization/palladium-catalyzed coupling.[J]. Acs Combinatorial Science, 2011, 13(5):501-510.