HPK1-IN-2 dihydrochloride

TargetMol
Product Code: TAR-T9017
Supplier: TargetMol
CodeSizePrice
TAR-T9017-1mg1mg£165.00
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TAR-T9017-5mg5mg£266.00
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Quantity:
TAR-T9017-10mg10mg£396.00
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Quantity:
TAR-T9017-25mg25mg£613.00
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Quantity:
TAR-T9017-50mg50mg£843.00
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Quantity:
TAR-T9017-100mg100mg£1,099.00
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Quantity:
TAR-T9017-500mg500mg£2,151.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
HPK1-IN-2 dihydrochloride is a potent and orally active inhibitor of hematopoietic progenitor kinase-1 (HPK1;IC50<0.05 μμ). It also inhibits Lck (0.05 μμ
CAS:
2056122-11-1
Formula:
C19H20N6OS
Molecular Weight:
380.47
Pathway:
Tyrosine Kinase/Adaptors; ; Angiogenesis
Purity:
0.9962
SMILES:
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2ccsc2[nH]c1=O
Target:
FLT; Src

References

Peter Brent Sampson, et al. Hpk1 inhibitors and methods of using same. WO2016205942A1.