Stafia-1

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TargetMol
Product Code: TAR-T9339
Supplier: TargetMol
CodeSizePrice
TAR-T9339-1mg1mg£133.00
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TAR-T9339-5mg5mg£229.00
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TAR-T9339-1mL1 mL * 10 mM (in DMSO)£254.00
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TAR-T9339-10mg10mg£332.00
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TAR-T9339-25mg25mg£515.00
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TAR-T9339-50mg50mg£710.00
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TAR-T9339-100mg100mg£946.00
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TAR-T9339-500mg500mg£1,854.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Stafia-1 is a potent STAT5a inhibitor ( IC50=22.2 μM). Stafia-1 displays high selectivity over STAT5b and other STAT family members.
CAS:
2582757-90-0
Formula:
C24H27O10P
Molecular Weight:
506.44
Pathway:
Stem Cells; JAK/STAT signaling
Purity:
0.9815
SMILES:
COC1=CC(C2=CC(OP(O)(O)=O)=CC(C3=CC(OC)=C(OC)C(OC)=C3)=C2)=CC(OC)=C1OC
Target:
STAT

References

Natarajan K, et al. Stafia-1: a STAT5a-Selective Inhibitor Developed via Docking-Based Screening of in Silico O-Phosphorylated Fragments. Chemistry. 2020;26(1):148-154.