Upidosin

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TargetMol
Product Code: TAR-T9762
Supplier: TargetMol
CodeSizePrice
TAR-T9762-5mg5mg£120.00
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Quantity:
TAR-T9762-1mL1 mL * 10 mM (in DMSO)£138.00
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Quantity:
TAR-T9762-10mg10mg£145.00
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Quantity:
TAR-T9762-25mg25mg£193.00
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Quantity:
TAR-T9762-50mg50mg£246.00
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Quantity:
TAR-T9762-100mg100mg£334.00
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Quantity:
TAR-T9762-200mg200mg£466.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Upidosin is a potential uroselective α1-adrenoceptor antagonist, α1a subtype Ki=0.34 nM, α1b subtype Ki=3.9 nM, α1d subtype Ki=1.5 nM, α2-adrenoceptor Ki=33.3 nM.
CAS:
152735-23-4
Formula:
C31H33N3O4
Molecular Weight:
511.61
Pathway:
Neuroscience; GPCR/G Protein
Purity:
0.9926
SMILES:
O=C(NCCCN1CCN(C=2C=CC=CC2OC)CC1)C3=CC=CC=4C(=O)C(=C(OC34)C=5C=CC=CC5)C
Target:
Adrenergic Receptor

References

Boschi D, et al. New potential uroselective NO-donor alpha1-antagonists. J Med Chem. 2003 Aug 14;46(17):3762-5.