Sarafotoxin S6c

TargetMol
Product Code: TAR-TP2120
Supplier: TargetMol
CodeSizePrice
TAR-TP2120-1mg1mg£521.00
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Quantity:
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Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Further Information

Bioactivity:
Highly selective ETB endothelin receptor agonist (Ki values are 0.29 and 28000 nM at ETB and ETA receptors respectively).
CAS:
121695-87-2
Formula:
C103H147N27O37S5
Molecular Weight:
2516
Purity:
0.98
SMILES:
0

References

Williams et al (1993) Characterization of cloned human endothelin receptors. Life Sci. 53 407 PMID: Matsuo et al (1997) Effects of sarafotoxin S6c on antidiuresis and NE overflow induced by stimulation of renal nerves in anesthetized dogs. J.Pharmacol.Exp.Ther. 280 905 PMID: Williams et al (1991) Sarafotoxin S6c: an agonist which distinguishes between endothelin receptor subtypes. Biochem.Biophys.Res.Commun. 175 556 PMID: Miasiro et al (1998) Distinct endothelin-B receptors mediate the effects of sarafotoxin S6c and IRL 1620 in the ileum. J.Cardiovasc.Pharmacol. 31 S175 PMID: