TargetMol

CP-809101 hydrochloride

Product Code:
 
TAR-T10871
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T10871-1mg1mg£97.00
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TAR-T10871-2mg2mg£107.00
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TAR-T10871-5mg5mg£131.00
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TAR-T10871-10mg10mg£164.00
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TAR-T10871-25mg25mg£278.00
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TAR-T10871-50mg50mg£455.00
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TAR-T10871-100mg100mg£621.00
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Further Information

Bioactivity:
CP-809101 hydrochloride is a potent and selective 5-HT2C receptor agonist (pEC50: 9.96/7.19/6.81 for human 5-HT2C/5-HT2B/5-HT2A receptors).
CAS:
1215721-40-6
Formula:
C15H18Cl2N4O
Molecular Weight:
341.24
Pathway:
GPCR/G Protein; Neuroscience
Purity:
0.9946
SMILES:
Cl.Clc1cccc(COc2cncc(n2)N2CCNCC2)c1
Target:
5-HT Receptor

References

1. Higgins GA, Silenieks LB, Lau W, et al. Evaluation of chemically diverse 5-HT2C receptor agonists on behaviours motivated by food and nicotine and on side effect profiles. Psychopharmacology (Berl). 2013 Apr;226(3):475-90. 2. Strong PV, Christianson JP, Loughridge AB, et al. 5-hydroxytryptamine 2C receptors in the dorsal striatum mediate stress-induced interference with negatively reinforced instrumental escape behavior. Neuroscience. 2011 Dec 1;197:132-44. doi: 10.1016/j.neuroscience.2011.09.041. Epub 2011 Sep 24. 3. Fletcher PJ, Tampakeras M, Sinyard J et al. Characterizing the effects of 5-HT(2C) receptor ligands on motor activity and feeding behaviour in 5-HT(2C) receptor knockout mice. Neuropharmacology. 2009 Sep;57(3):259-67. doi: 10.1016/j.neuropharm.2009.05.011. 4. Siuciak JA, Chapin DS, McCarthy SA, et al. CP-809,101, a selective 5-HT2C agonist, shows activity in animal models of antipsychotic activity. Neuropharmacology. 2007 Feb;52(2):279-90.