Telotristat ethyl

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TargetMol
Product Code: TAR-T11897
Supplier: TargetMol
CodeSizePrice
TAR-T11897-1mg1mg£103.00
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TAR-T11897-2mg2mg£118.00
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TAR-T11897-5mg5mg£148.00
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TAR-T11897-1mL1 mL * 10 mM (in DMSO)£169.00
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TAR-T11897-10mg10mg£214.00
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TAR-T11897-25mg25mg£310.00
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TAR-T11897-50mg50mg£426.00
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TAR-T11897-100mg100mg£595.00
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TAR-T11897-500mg500mg£1,187.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Telotristat ethyl is a orally-delivered inhibitor of tryptophan hydroxylase that reduces serotonin production.
CAS:
1033805-22-9
Formula:
C27H26ClF3N6O3
Molecular Weight:
574.99
Pathway:
Metabolism
Purity:
0.9972
SMILES:
CCOC(=O)[C@@H](N)Cc1ccc(cc1)-c1cc(O[C@H](c2ccc(Cl)cc2-n2ccc(C)n2)C(F)(F)F)nc(N)n1
Target:
Hydroxylase

References

1. Tamas Oravecz, et al. LX1606 (aka LX1032), a Novel Inhibitor of Serotonin Synthesis, Alleviates Development of Inflammatory Bowel Disease in a Preclinical Model. 2. Margolis, K.G., et al., Pharmacological reduction of mucosal but not neuronal serotonin opposes inflammation in mouse intestine. Gut, 2013.