(±)-Enitociclib

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TargetMol
Product Code: TAR-T13467
Supplier: TargetMol
CodeSizePrice
TAR-T13467-1mg1mg£122.00
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TAR-T13467-2mg2mg£144.00
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TAR-T13467-1mL1 mL * 10 mM (in DMSO)£181.00
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TAR-T13467-5mg5mg£197.00
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Quantity:
TAR-T13467-10mg10mg£264.00
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Quantity:
TAR-T13467-25mg25mg£389.00
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TAR-T13467-50mg50mg£544.00
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TAR-T13467-100mg100mg£760.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
(?)-BAY-1251152 is a racemic mixture of BAY-1251152. BAY-1251152 is highly selective inhibitor of PTEF/CDK9.
CAS:
1610358-53-6
Formula:
C19H18F2N4O2S
Molecular Weight:
404.44
Pathway:
Cell Cycle/Checkpoint
Purity:
0.9946
SMILES:
COc1cc(F)ccc1-c1cc(Nc2cc(CS(C)(=N)=O)ccn2)ncc1F
Target:
CDK

References

1. Luecking, et al. Identification of potent and highly selective PTEFb inhibitor BAY 1251152 for the treatment of cancer: from p.o. to i.v. application via scaffold hops [abstract]. In: Proceedings of the American Association for Cancer Research Annual Meeting 2017; 2017 Apr 1-5; Washington, DC. Philadelphia (PA): AACR; Cancer Res 2017;77(13 Suppl):Abstract nr 984. doi:10.1158/1538-7445.AM2017-984