Taselisib

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TargetMol
Product Code: TAR-T1999
Supplier: TargetMol
CodeSizePrice
TAR-T1999-2mg2mg£101.00
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TAR-T1999-1mL1 mL * 10 mM (in DMSO)£119.00
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TAR-T1999-5mg5mg£119.00
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TAR-T1999-10mg10mg£145.00
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Quantity:
TAR-T1999-25mg25mg£198.00
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TAR-T1999-50mg50mg£237.00
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TAR-T1999-100mg100mg£367.00
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TAR-T1999-200mg200mg£511.00
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TAR-T1999-500mg500mg£781.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Taselisib is an orally bioavailable inhibitor of the class I phosphatidylinositol 3-kinase (PI3K) alpha isoform (PIK3CA), with potential antineoplastic activity.
CAS:
1282512-48-4
Formula:
C24H28N8O2
Molecular Weight:
460.542
Pathway:
PI3K/Akt/mTOR signaling; Metabolism
Purity:
0.9962
SMILES:
CC(C)n1nc(C)nc1-c1cn2CCOc3cc(ccc3-c2n1)-c1cnn(c1)C(C)(C)C(N)=O
Target:
PI3K; Carbonic Anhydrase

References

1. Ndubaku CO, et al. J Med Chem, 2013, 56(11), 4597-4610.