LY2409881 trihydrochloride

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TargetMol
Product Code: TAR-T2081
Supplier: TargetMol
CodeSizePrice
TAR-T2081-1mg1mg£107.00
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TAR-T2081-2mg2mg£122.00
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TAR-T2081-5mg5mg£149.00
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TAR-T2081-1mL1 mL * 10 mM (in DMSO)£182.00
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TAR-T2081-10mg10mg£213.00
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TAR-T2081-25mg25mg£354.00
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TAR-T2081-50mg50mg£510.00
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TAR-T2081-100mg100mg£703.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
LY2409881 trihydrochloride is a novel specific inhibitor of IKK2 (IC50: 30 nM); IC50 for IKK1 and other common kinases is at least one log higher.
CAS:
946518-60-1
Formula:
C24H32Cl4N6OS
Molecular Weight:
594.42
Pathway:
Apoptosis; NF-κb
Purity:
0.98
SMILES:
Cl.Cl.Cl.CN1CCN(CCCNc2ncc(Cl)c(n2)-c2cc3c(cccc3s2)C(=O)NC2CC2)CC1
Target:
Apoptosis; IκB/IKK

References

1. Deng C, et al. Clin Cancer Res. 2015, 21(1):134-145.