CCT 137690

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TargetMol
Product Code: TAR-T2611
Supplier: TargetMol
CodeSizePrice
TAR-T2611-2mg2mg£111.00
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TAR-T2611-5mg5mg£128.00
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TAR-T2611-1mL1 mL * 10 mM (in DMSO)£140.00
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TAR-T2611-10mg10mg£145.00
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TAR-T2611-25mg25mg£216.00
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TAR-T2611-50mg50mg£334.00
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TAR-T2611-100mg100mg£480.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
CCT 137690 is a highly specific and oral-available aurora kinase inhibitor, for aurora A(IC50=15 nM ), B(IC50=25 nM) and C(IC50=19 nM).
CAS:
1095382-05-0
Formula:
C26H31BrN8O
Molecular Weight:
551.493
Pathway:
Chromatin/Epigenetic; Cell Cycle/Checkpoint; Apoptosis
Purity:
0.9851
SMILES:
CN1CCN(CC1)c1ccc(cc1)-c1nc2c(N3CCN(Cc4cc(C)on4)CC3)c(Br)cnc2[nH]1
Target:
Apoptosis; Aurora Kinase

References

1. Bavetsias V, et al. J Med Chem, 2010, 53(14), 5213-5228. 2. Faisal A, et al. Mol Cancer Ther, 2011, 10(11), 2115-2123. 3. Moore AS, et al. ASH Annu Meeting Abstr, 2010, 116, Abstr 3289.