CUDC-101

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TargetMol
Product Code: TAR-T3108
Supplier: TargetMol
CodeSizePrice
TAR-T3108-5mg5mg£105.00
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TAR-T3108-1mL1 mL * 10 mM (in DMSO)£109.00
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TAR-T3108-10mg10mg£132.00
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TAR-T3108-25mg25mg£172.00
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TAR-T3108-50mg50mg£237.00
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TAR-T3108-100mg100mg£367.00
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TAR-T3108-500mg500mg£781.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CUDC-101 is a potent inhibitor of HDAC, EGFR and HER2 with IC50s of 4.4, 2.4 and 15.7 nM, respectively.
CAS:
1012054-59-9
Formula:
C24H26N4O4
Molecular Weight:
434.496
Pathway:
DNA Damage/DNA Repair; Tyrosine Kinase/Adaptors; JAK/STAT signaling; Chromatin/Epigenetic; Angiogenesis
Purity:
0.9912
SMILES:
COc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCCCCCC(=O)NO
Target:
EGFR; HER; HDAC

References

1. Cai X, et al. J Med Chem, 2010, 53(5), 2000-2009. 2. Lai CJ, et al. Cancer Res, 2010, 70(9), 3647-3656.