CRT0273750

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TargetMol
Product Code: TAR-T31101
Supplier: TargetMol
CodeSizePrice
TAR-T31101-1mg1mg£115.00
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TAR-T31101-2mg2mg£134.00
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TAR-T31101-5mg5mg£168.00
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TAR-T31101-1mL1 mL * 10 mM (in DMSO)£179.00
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TAR-T31101-10mg10mg£229.00
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TAR-T31101-25mg25mg£430.00
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TAR-T31101-50mg50mg£600.00
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TAR-T31101-100mg100mg£825.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
CRT0273750 regulates plasma LPA levels and is suitable for in vivo studies. CRT0273750 is an autotaxin (ATX) inhibitor with IC50 of 0.014 μM.
CAS:
1979939-16-6
Formula:
C25H22ClF3N4O2
Molecular Weight:
502.92
Pathway:
Metabolism
Purity:
0.9949
SMILES:
C[C@H](NC(=O)CCc1nc2cccnc2n1Cc1ccc(OC(F)(F)F)cc1)c1ccc(Cl)cc1
Target:
PDE

References

1. Shah P, et al. Discovery of potent inhibitors of the lysophospholipase autotaxin. Bioorg Med Chem Lett. 2016 Nov 15;26(22):5403-5410.