K858 (Racemic)

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TargetMol
Product Code: TAR-T3120
Supplier: TargetMol
CodeSizePrice
TAR-T3120-5mg5mg£102.00
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Quantity:
TAR-T3120-1mL1 mL * 10 mM (in DMSO)£105.00
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Quantity:
TAR-T3120-10mg10mg£128.00
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Quantity:
TAR-T3120-25mg25mg£198.00
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Quantity:
TAR-T3120-50mg50mg£302.00
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Quantity:
TAR-T3120-100mg100mg£490.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
K858 is a selective mitotic kinesin Eg5 inhibitor which acts in an ATP-noncompetitive manner.
CAS:
72926-24-0
Formula:
C13H15N3O2S
Molecular Weight:
277.34
Pathway:
Cytoskeletal Signaling; Apoptosis
Purity:
0.995
SMILES:
CC(=O)NC1=NN(C(C)=O)C(C)(S1)c1ccccc1
Target:
Apoptosis; Kinesin

References

1. Nakai R, et al. Y Res. 2009 May 1;69(9):3901-9. 2. Indorato RL, et al. Biochem Pharmacol. 2013 Nov 15;86(10):1441-51.