GRA Ex-25

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TargetMol
Product Code: TAR-T3422
Supplier: TargetMol
CodeSizePrice
TAR-T3422-1mg1mg£116.00
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TAR-T3422-2mg2mg£136.00
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TAR-T3422-5mg5mg£185.00
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TAR-T3422-1mL1 mL * 10 mM (in DMSO)£228.00
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TAR-T3422-10mg10mg£244.00
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TAR-T3422-25mg25mg£425.00
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TAR-T3422-50mg50mg£592.00
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TAR-T3422-100mg100mg£814.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GRA-Ex-25 is an inhibitor of glucagon receptor.
CAS:
307983-31-9
Formula:
C29H36F3N3O5
Molecular Weight:
563.618
Pathway:
GPCR/G Protein
Purity:
0.982
SMILES:
CC(C)(C)C1CCC(CC1)N(Cc1ccc(cc1)C(=O)NCCC(O)=O)C(=O)Nc1ccc(OC(F)(F)F)cc1
Target:
Glucagon Receptor

References

Lau J, et al. New beta-alanine derivatives are orally available glucagon receptor antagonists. J Med Chem. 2007 Jan 11;50(1):113-28. Kurukulasuriya R, et al. Biaryl amide glucagon receptor antagonists. Bioorg Med Chem Lett. 2004 May 3;14(9):2047-50. Li Y, Zhou X, Cheng C, et al.Gut AstA mediates sleep deprivation-induced energy wasting in Drosophila.Cell Discovery.2023, 9(1): 49.