EED226

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TargetMol
Product Code: TAR-T3458
Supplier: TargetMol
CodeSizePrice
TAR-T3458-2mg2mg£98.00
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Quantity:
TAR-T3458-1mL1 mL * 10 mM (in DMSO)£109.00
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Quantity:
TAR-T3458-5mg5mg£109.00
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Quantity:
TAR-T3458-10mg10mg£132.00
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Quantity:
TAR-T3458-25mg25mg£172.00
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Quantity:
TAR-T3458-50mg50mg£237.00
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Quantity:
TAR-T3458-100mg100mg£367.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
EED226 is a potent, selective, and orally bioavailable embryonic ectoderm development (EED) inhibitor with an IC50 of 22 nM.
CAS:
2083627-02-3
Formula:
C17H15N5O3S
Molecular Weight:
369.4
Pathway:
Chromatin/Epigenetic
Purity:
0.9966
SMILES:
CS(=O)(=O)c1ccc(cc1)-c1cnc(NCc2ccco2)n2cnnc12
Target:
DNA Methyltransferase; Histone Methyltransferase

References

Cancer Discov. 2017, 7(4):OF8. doi: 10.1158/2159-8290.CD-RW2017-030. Qi W, et al. Nat Chem Biol. 2017, 13(4):381-388. Y Huang, et al. J Med Chem. 60 (6):2215-2226.