U93631

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TargetMol
Product Code: TAR-T3644
Supplier: TargetMol
CodeSizePrice
TAR-T3644-5mg5mg£102.00
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Quantity:
TAR-T3644-1mL1 mL * 10 mM (in DMSO)£105.00
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Quantity:
TAR-T3644-10mg10mg£122.00
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Quantity:
TAR-T3644-25mg25mg£173.00
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Quantity:
TAR-T3644-50mg50mg£230.00
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Quantity:
TAR-T3644-100mg100mg£367.00
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Quantity:
TAR-T3644-500mg500mg£768.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GABAA receptor antagonist that binds the picrotoxin site and stabilizes the inactive form of the channel via allosteric interaction. Accelerates the decay of GABA-induced Cl- currents with little effect on peak amplitude. Also inhibits 5-HT3A receptors via a similar mechanism.
CAS:
152273-12-6
Formula:
C17H21N3O2
Molecular Weight:
299.374
Pathway:
Neuroscience; Membrane transporter/Ion channel
Purity:
0.9997
SMILES:
CC(C)(C)OC(=O)c1ncn-2c1C(C)(C)Nc1ccccc-21
Target:
GABA Receptor

References

Dillon,GH et al. Mol Pharmacol. 1993 Oct;44(4):860-5.