PF-CBP1

TargetMol
Product Code: TAR-T3973
Supplier: TargetMol
CodeSizePrice
TAR-T3973-1mg1mg£100.00
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TAR-T3973-2mg2mg£111.00
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TAR-T3973-1mL1 mL * 10 mM (in DMSO)£121.00
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Quantity:
TAR-T3973-5mg5mg£121.00
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TAR-T3973-10mg10mg£159.00
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TAR-T3973-25mg25mg£244.00
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TAR-T3973-50mg50mg£385.00
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TAR-T3973-100mg100mg£538.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

1 / 1

Further Information

Bioactivity:
PF-CBP1 HCl is a highly selective inhibitor of the bromodomain of CREB-binding protein(CREBBP). It inhibits CREBBP (IC50: 125 nM) and p300 bromodomains (IC50: 363 nM).
CAS:
1962928-21-7
Formula:
C29H36N4O3
Molecular Weight:
488.632
Pathway:
Chromatin/Epigenetic
Purity:
0.9991
SMILES:
CCCOc1ccc(CCc2nc3cc(ccc3n2CCN2CCOCC2)-c2c(C)noc2C)cc1
Target:
Epigenetic Reader Domain

References

Eugene L, et al. Chem Biol. 2015, 22(12):1588-1596.