WDR5-0103 hydrochloride[890190-22-4(free base)]

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TargetMol
Product Code: TAR-T5140
Supplier: TargetMol
CodeSizePrice
TAR-T5140-1mg1mg£100.00
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TAR-T5140-2mg2mg£111.00
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TAR-T5140-5mg5mg£124.00
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Quantity:
TAR-T5140-10mg10mg£168.00
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Quantity:
TAR-T5140-25mg25mg£246.00
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Quantity:
TAR-T5140-50mg50mg£375.00
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TAR-T5140-100mg100mg£452.00
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TAR-T5140-200mg200mg£629.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
WDR5-0103 is an effective and specific WD repeat-containing protein 5 (WDR5) antagonist (Kd: 450 nM).
CAS:
T5140
Formula:
C21H26ClN3O4
Molecular Weight:
419.9
Pathway:
JAK/STAT signaling; Angiogenesis; Chromatin/Epigenetic; Stem Cells
Purity:
0.9981
SMILES:
Cl.COC(=O)c1ccc(N2CCN(C)CC2)c(NC(=O)c2cccc(OC)c2)c1
Target:
JAK

References

Senisterra G, et al. Small-molecule inhibition of MLL activity by disruption of its interaction with WDR5. Biochem J. 2013 Jan 1;449(1):151-159.