MC180295

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TargetMol
Product Code: TAR-T5533
Supplier: TargetMol
CodeSizePrice
TAR-T5533-1mg1mg£139.00
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TAR-T5533-2mg2mg£169.00
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TAR-T5533-5mg5mg£249.00
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TAR-T5533-1mL1 mL * 10 mM (in DMSO)£266.00
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Quantity:
TAR-T5533-10mg10mg£335.00
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Quantity:
TAR-T5533-25mg25mg£519.00
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TAR-T5533-50mg50mg£702.00
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TAR-T5533-100mg100mg£970.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
MC180295 is a novel potent, highly selective CDK9 inhibitor (IC50: 5 nM), displays >22-fold selectivity over other CDKs.
CAS:
2237942-08-2
Formula:
C17H18N4O3S
Molecular Weight:
358.42
Pathway:
Cell Cycle/Checkpoint
Purity:
0.98
SMILES:
Nc1nc(N[C@H]2CC3CCC2C3)sc1C(=O)c1ccccc1[N+]([O-])=O
Target:
CDK

References

Zhang H, et al. Targeting CDK9 Reactivates Epigenetically Silenced Genes in Cancer. Cell. 2018 Nov 15;175(5):1244-1258.e26.