GSK8612

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TargetMol
Product Code: TAR-T5540
Supplier: TargetMol
CodeSizePrice
TAR-T5540-1mg1mg£102.00
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TAR-T5540-2mg2mg£114.00
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TAR-T5540-5mg5mg£138.00
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TAR-T5540-1mL1 mL * 10 mM (in DMSO)£148.00
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TAR-T5540-10mg10mg£177.00
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TAR-T5540-25mg25mg£252.00
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TAR-T5540-50mg50mg£389.00
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TAR-T5540-100mg100mg£550.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
GSK8612 is a highly selective and potent inhibitor of Tank-binding Kinase-1 (TBK1, pIC50: 6.8) .
CAS:
2361659-62-1
Formula:
C17H17BrF3N7O2S
Molecular Weight:
520.33
Pathway:
NF-κb
Purity:
0.998
SMILES:
Cc1nn(CC(F)(F)F)cc1Nc1ncc(Br)c(NCc2ccc(cc2)S(N)(=O)=O)n1
Target:
IκB/IKK

References

Thomson DW, et al. Discovery of GSK8612, a Highly Selective and Potent TBK1 Inhibitor. ACS Med Chem Lett. 2019 Mar 11;10(5):780-785.