Entospletinib

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TargetMol
Product Code: TAR-T6101
Supplier: TargetMol
CodeSizePrice
TAR-T6101-1mg1mg£96.00
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TAR-T6101-2mg2mg£107.00
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TAR-T6101-5mg5mg£130.00
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TAR-T6101-1mL1 mL * 10 mM (in DMSO)£136.00
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TAR-T6101-10mg10mg£149.00
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TAR-T6101-25mg25mg£213.00
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TAR-T6101-50mg50mg£289.00
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TAR-T6101-100mg100mg£422.00
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TAR-T6101-200mg200mg£592.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
Entospletinib ?IC50= 7.7 nM?is a specific Syk inhibitor, which is orally bioavailable.
CAS:
1229208-44-9
Formula:
C23H21N7O
Molecular Weight:
411.469
Pathway:
Tyrosine Kinase/Adaptors; Angiogenesis
Purity:
0.9951
SMILES:
C1CN(CCO1)c1ccc(Nc2nc(cn3ccnc23)-c2ccc3cn[nH]c3c2)cc1
Target:
Syk

References

J Med Chem. 2014, 57(9), 3856-3873. Burke RT, et al. Oncotarget. 2014, 5(4), 908-915.