Darapladib

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TargetMol
Product Code: TAR-T6109
Supplier: TargetMol
CodeSizePrice
TAR-T6109-1mg1mg£106.00
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TAR-T6109-2mg2mg£122.00
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TAR-T6109-5mg5mg£148.00
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TAR-T6109-1mL1 mL * 10 mM (in DMSO)£196.00
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TAR-T6109-10mg10mg£209.00
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TAR-T6109-25mg25mg£349.00
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TAR-T6109-50mg50mg£523.00
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TAR-T6109-100mg100mg£702.00
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TAR-T6109-500mg500mg£1,348.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
Darapladib(IC50=0.25 nM) is a substituted pyrimidone with inhibitory activity towards lipoprotein-associated phospholipase-A2 (Lp-PLA2).
CAS:
356057-34-6
Formula:
C36H38F4N4O2S
Molecular Weight:
666.78
Pathway:
Metabolism
Purity:
0.9985
SMILES:
CCN(CC)CCN(Cc1ccc(cc1)-c1ccc(cc1)C(F)(F)F)C(=O)Cn1c2CCCc2c(=O)nc1SCc1ccc(F)cc1
Target:
Phospholipase

References

Blackie JA, et al. Bioorg Med Chem Lett. 2003, 13(6), 1067-1070. Wilensky RL, et al. Nat Med. 2008, 14(10), 1059-1066. Acharya NK, et al. J Alzheimers Dis. 2013, 35(1), 179-198.