AMG-208

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TargetMol
Product Code: TAR-T6260
Supplier: TargetMol
CodeSizePrice
TAR-T6260-1mg1mg£103.00
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TAR-T6260-2mg2mg£115.00
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Quantity:
TAR-T6260-5mg5mg£148.00
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TAR-T6260-10mg10mg£189.00
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Quantity:
TAR-T6260-25mg25mg£285.00
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TAR-T6260-50mg50mg£430.00
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TAR-T6260-100mg100mg£590.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
AMG 208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.
CAS:
1002304-34-8
Formula:
C22H17N5O2
Molecular Weight:
383.411
Pathway:
Metabolism; Tyrosine Kinase/Adaptors
Purity:
0.9913
SMILES:
COc1ccc2c(OCc3nnc4ccc(nn34)-c3ccccc3)ccnc2c1
Target:
P45; c-Met/HGFR

References

Liu X, et al. Trends Mol Med. 2010,16(1), 37-45. Boezio AA, et al. Bioorg Med Chem Lett. 2009, 19(22), 6307-6312. Albrecht BK, et al. J Med Chem. 2008, 51(10), 2879-2882.