BMS-378806

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TargetMol
Product Code: TAR-T6418
Supplier: TargetMol
CodeSizePrice
TAR-T6418-1mg1mg£107.00
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TAR-T6418-2mg2mg£121.00
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TAR-T6418-5mg5mg£168.00
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TAR-T6418-1mL1 mL * 10 mM (in DMSO)£177.00
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TAR-T6418-10mg10mg£229.00
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TAR-T6418-25mg25mg£401.00
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TAR-T6418-50mg50mg£574.00
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TAR-T6418-100mg100mg£788.00
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TAR-T6418-500mg500mg£1,508.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
BMS-378806 selectively inhibits the binding of HIV-1 gp120 to the CD4 receptor with EC50 of 0.85-26.5 nM in virus.
CAS:
357263-13-9
Formula:
C22H22N4O4
Molecular Weight:
406.442
Pathway:
Immunology/Inflammation; Microbiology/Virology; Proteases/Proteasome
Purity:
0.98
SMILES:
COc1ccnc2[nH]cc(C(=O)C(=O)N3CCN(C[C@H]3C)C(=O)c3ccccc3)c12
Target:
gp12/CD4; HIV Protease

References

Guo Q, et al, J Virol, 2003, 77(19), 10528-10536. Yang Z, et al, Biopharm Drug Dispos, 2005, 26(9) Wang T, et al, J Med Chem, 2003, 46(20), 4236-4239.