CPI-637

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TargetMol
Product Code: TAR-T6811
Supplier: TargetMol
CodeSizePrice
TAR-T6811-1mg1mg£98.00
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TAR-T6811-2mg2mg£108.00
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TAR-T6811-1mL1 mL * 10 mM (in DMSO)£128.00
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TAR-T6811-5mg5mg£128.00
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TAR-T6811-10mg10mg£152.00
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TAR-T6811-25mg25mg£250.00
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TAR-T6811-50mg50mg£389.00
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TAR-T6811-100mg100mg£550.00
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TAR-T6811-500mg500mg£1,083.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
CPI-637 is a selective and cell-active benzodiazepinone CBP/EP300 bromodomain inhibitor.
CAS:
1884712-47-3
Formula:
C22H22N6O
Molecular Weight:
386.459
Pathway:
Chromatin/Epigenetic
Purity:
0.9991
SMILES:
C[C@@H]1CC(=O)Nc2cccc(-c3ccc4n(C)nc(-c5cnn(C)c5)c4c3)c2N1
Target:
Epigenetic Reader Domain; Histone Acetyltransferase

References

Wang X, Xie Q, Ji Y, et al.Targeting KRAS-mutant stomach/colorectal tumors by disrupting the ERK2-p53 complex.Cell Reports.2023, 42(1): 111972. Taylor AM, et al. ACS Med Chem Lett. 2016, 7(5):531-6. Lang J Y, Wang X, Xie Q, et al. Targeting KRAS-mutant stomach/colorectal tumours by disrupting the ERK2-p53 complex[J]. bioRxiv. 2020