Oclacitinib maleate

TargetMol
Product Code: TAR-T6914
Supplier: TargetMol
CodeSizePrice
TAR-T6914-1mg1mg£97.00
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TAR-T6914-2mg2mg£107.00
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TAR-T6914-5mg5mg£128.00
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TAR-T6914-1mL1 mL * 10 mM (in DMSO)£133.00
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TAR-T6914-10mg10mg£152.00
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TAR-T6914-25mg25mg£213.00
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TAR-T6914-50mg50mg£300.00
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TAR-T6914-100mg100mg£456.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Further Information

Bioactivity:
Oclacitinib is a novel inhibitor of JAK family members with IC50 ranging from 10 to 99 nM and JAK1-dependent cytokines with IC50 ranging from 36 to 249 nM, which did not inhibit a panel of 38 non-JAK kinases.
CAS:
1640292-55-2
Formula:
C19H27N5O6S
Molecular Weight:
453.51
Pathway:
Chromatin/Epigenetic; Angiogenesis; Tyrosine Kinase/Adaptors; JAK/STAT signaling; Stem Cells
Purity:
0.9917
SMILES:
OC(=O)C=C/C(O)=O.CNS(=O)(=O)C[C@H]1CC[C@@H](CC1)N(C)c1ncnc2[nH]ccc12
Target:
Tyrosine Kinases; JAK

References

Cosgrove SB, et al. Vet Dermatol. 2013, 24(5):479-e114. Gonzales AJ, et al. J Vet Pharmacol Ther. 2014, 37(4):317-324.