G15

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TargetMol
Product Code: TAR-T7389
Supplier: TargetMol
CodeSizePrice
TAR-T7389-1mg1mg£97.00
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TAR-T7389-5mg5mg£131.00
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TAR-T7389-1mL1 mL * 10 mM (in DMSO)£137.00
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TAR-T7389-10mg10mg£171.00
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TAR-T7389-25mg25mg£254.00
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TAR-T7389-50mg50mg£383.00
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TAR-T7389-100mg100mg£540.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
G15 is a cell-permeable non-steroidal antagonist of GPER (Ki = 20 nM)
CAS:
1161002-05-6
Formula:
C19H16BrNO2
Molecular Weight:
370.246
Pathway:
Endocrinology/Hormones
Purity:
0.98
SMILES:
Brc1cc2OCOc2cc1[C@@H]1Nc2ccccc2[C@@H]2C=CC[C@H]12
Target:
Estrogen Receptor/ERR

References

Bai L Y , Weng J R , Hu J L , et al. G15, a GPR30 antagonist, induces apoptosis and autophagy in human oral squamous carcinoma cells[J]. Chemico-Biological Interactions, 2013, 206(2):375-384. Nayak T K , Bologa C G , Leitao A , et al. In vivo effects of a GPR30 antagonist[J]. Nature Chemical Biology, 2009, 5(6):421-427.