TargetMol

GW284543

Product Code:
 
TAR-T7610
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T7610-1mg1mg£95.00
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TAR-T7610-5mg5mg£128.00
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TAR-T7610-1mL1 mL * 10 mM (in DMSO)£134.00
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TAR-T7610-10mg10mg£161.00
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TAR-T7610-25mg25mg£242.00
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TAR-T7610-50mg50mg£369.00
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Quantity:
TAR-T7610-100mg100mg£517.00
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Quantity:
TAR-T7610-500mg500mg£1,050.00
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Quantity:
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
GW284543 is a selective inhibitor of MEK5 .
CAS:
790186-68-4
Formula:
C23H20N2O3
Molecular Weight:
372.424
Pathway:
MAPK
Purity:
0.9964
SMILES:
COc1cc2nccc(Nc3cccc(Oc4ccccc4)c3)c2cc1OC
Target:
MEK

References

Vaseva AV, Blake DR, Gilbert TSK,et al.KRAS Suppression-Induced Degradation of MYC Is Antagonized by a MEK5-ERK5 Compensatory Mechanism[J].Cancer Cell. 2018 Nov 12;34(5):807-822.e7.