Nitecapone

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TargetMol

Product Code: TAR-T7831

Product Group: Inhibitors and Activators

Supplier: TargetMol

Code	Size	Price

TAR-T7831-1mg

1mg

£125.00

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Quantity:

TAR-T7831-2mg

2mg

£149.00

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Quantity:

TAR-T7831-5mg

5mg

£209.00

Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.

Quantity:

TAR-T7831-10mg

10mg

£302.00

Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.

Quantity:

TAR-T7831-25mg

25mg

£463.00

Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.

Quantity:

TAR-T7831-50mg

50mg

£621.00

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Quantity:

TAR-T7831-100mg

100mg

£830.00

Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.

Quantity:

Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO

Shipping:

cool pack

Storage:

-20℃

Images

1 / 1

Documents

Further Information

Bioactivity:

Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)

CAS:

116313-94-1

Formula:

C12H11NO6

Molecular Weight:

265.221

Pathway:

; Metabolism

Purity:

0.99

SMILES:

CC(=O)C(=Cc1cc(O)c(O)c(c1)[N+]([O-])=O)C(C)=O

Target:

Transferase

References

Salmela K S , Roine R P , H??K-Nikanne J , et al. Effect of Bismuth and Nitecapone on Acetaldehyde Production by Helicobacter pylori[J]. Scandinavian Journal of Gastroenterology, 1994, 29(6):528-531. P.T. M?nnist?, Kaakkola S . Catechol-O-methyltransferase (COMT): Biochemistry, molecular biology, pharmacology, and clinical efficacy of the new selective COMT inhibitors[J]. Pharmacological Reviews, 2000, 51(4):593-628. Inhibitors of catechol?O?methyltransferase sensitize mice to pain[J]. British Journal of Pharmacology, 2010, 161(7).