PW0787

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TargetMol
Product Code: TAR-T9452
Supplier: TargetMol
CodeSizePrice
TAR-T9452-1mg1mg£111.00
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TAR-T9452-2mg2mg£130.00
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TAR-T9452-5mg5mg£168.00
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Quantity:
TAR-T9452-1mL1 mL * 10 mM (in DMSO)£189.00
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TAR-T9452-10mg10mg£230.00
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Quantity:
TAR-T9452-25mg25mg£402.00
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TAR-T9452-50mg50mg£568.00
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TAR-T9452-100mg100mg£777.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
PW0787 is a potent, selective, orally active, and brain-penetrant GPR52 agonist (EC50=135 nM).
CAS:
2624131-45-7
Formula:
C23H20F4N4O2
Molecular Weight:
460.433
Pathway:
Endocrinology/Hormones; GPCR/G Protein
Purity:
0.9852
SMILES:
OCCNC(=O)c1cccc2N(CCc12)c1cc(Cc2cc(F)cc(c2)C(F)(F)F)ncn1
Target:
GPR

References

Wang P, et al. Discovery of Potent and Brain-Penetrant GPR52 Agonist that Suppresses Psychostimulant Behavior. J Med Chem. 2020;63(22):13951-13972.