TargetMol

GPR40/FFAR1 modulator 1

Product Code:
 
TAR-T11458
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T11458-5mg5mg£107.00
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TAR-T11458-10mg10mg£130.00
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TAR-T11458-1mL1 mL * 10 mM (in DMSO)£138.00
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TAR-T11458-25mg25mg£177.00
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TAR-T11458-50mg50mg£244.00
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TAR-T11458-100mg100mg£351.00
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Further Information

Bioactivity:
GPR40/FFAR1 modulator 1 is an agonist and an allosteric modulator for Gq-coupled free fatty acid receptor 1 (GPR40/FFAR1).
CAS:
874755-26-7
Formula:
C21H19N5O3
Molecular Weight:
389.415
Pathway:
GPCR/G Protein; Endocrinology/Hormones
Purity:
0.9972
SMILES:
Cc1ccccc1Nc1nc(N)nc(COc2ccc3c(C)cc(=O)oc3c2)n1
Target:
GPR

References

1. L?ckmann M, et al. Molecular dynamics-guided discovery of an ago-allosteric modulator for GPR40/FFAR1. Proc Natl Acad Sci U S A. 2019 Apr 2;116(14):7123-7128.