TargetMol

PF-06726304 acetate

Product Code:
 
TAR-T12428
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12428-5mg5mg£1,251.00
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TAR-T12428-50mg50mg£2,464.00
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Quantity:
TAR-T12428-100mg100mg£3,283.00
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This product comes from: United States.
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Further Information

Bioactivity:
PF-06726304 acetate is a selective inhibitor of EZH2, with robust antitumor growth activity.
CAS:
2080306-28-9
Formula:
C24H25Cl2N3O5
Molecular Weight:
506.38
Pathway:
Chromatin/Epigenetic
Purity:
0.98
SMILES:
CC(O)=O.Cc1noc(C)c1-c1cc(Cl)c2CCN(Cc3c(C)cc(C)[nH]c3=O)C(=O)c2c1Cl
Target:
Histone Methyltransferase

References

1. Kung PP, et al. Design and Synthesis of Pyridone-Containing 3,4-Dihydroisoquinoline-1(2H)-ones as a Novel Class of Enhancer of Zeste Homolog 2 (EZH2) Inhibitors. J Med Chem. 2016 Sep 22;59(18):8306-25.