TargetMol

PI3Kdelta inhibitor 1

Product Code:
 
TAR-T12461
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12461-5mg5mg£850.00
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TAR-T12461-50mg50mg£1,661.00
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Quantity:
TAR-T12461-100mg100mg£2,079.00
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This product comes from: United States.
Typical lead time: 10-14 working days.
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Further Information

Bioactivity:
PI3Kdelta inhibitor 1 is a potent, selective and orally available inhibitor of PI3Kδ with an IC50 of 1.3 nM.
CAS:
2242109-74-4
Formula:
C27H38N6O5S
Molecular Weight:
558.7
Pathway:
PI3K/Akt/mTOR signaling
Purity:
0.98
SMILES:
COc1ncc(cc1NS(C)(=O)=O)-c1cc(OC[C@@H]2CCCN(CCC3CCOCC3)C2)c2cnn(C)c2n1
Target:
PI3K

References

1. Hamajima T, et al. Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3K? inhibitor. Bioorg Med Chem. 2018 Aug 7;26(14):3917-3924.