Pinacidil
Code | Size | Price |
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TAR-T12478L-5mg | 5mg | £104.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T12478L-1mL | 1 mL * 10 mM (in DMSO) | £107.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T12478L-10mg | 10mg | £117.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T12478L-25mg | 25mg | £148.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
TAR-T12478L-50mg | 50mg | £203.00 | |||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||||
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here. |
Quantity:
Prices exclude any Taxes / VAT
Overview
Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃
Images
Documents
Further Information
Bioactivity:
Pinardil (P-1134, S-1230) is a guanidine that opens potassium channels and directly dilates peripheral blood vessels in small arteries, lowering blood pressure and peripheral resistance and producing fluid retention.
CAS:
60560-33-0
Formula:
C13H19N5
Molecular Weight:
245.33
Pathway:
Membrane transporter/Ion channel
Purity:
0.98
SMILES:
CC(C)(C)C(N/C(NC1=CC=NC=C1)=N/C#N)C
Target:
Potassium Channel
References
1. Friedel HA, Brogden RN. Pinacidil. A review of its pharmacodynamic and pharmacokinetic properties, and therapeutic potential in the treatment of hypertension. Drugs. 1990 Jun;39(6):929-67. Review. PubMed PMID: 2196168.
2. Ahnfelt-R?nne I. Pinacidil. Preclinical investigations. Drugs. 1988;36 Suppl 7:4-9. Review. PubMed PMID: 3076134.
3. Cohen ML, Kurz KD. Pinacidil-induced vascular relaxation: comparison to other vasodilators and to classical mechanisms of vasodilation. J Cardiovasc Pharmacol. 1988;12 Suppl 2:S5-9. PubMed PMID: 2466179.
4. Zushida K, Onodera K, Kamei J. Effect of diabetes on pinacidil-induced antinociception in mice. Eur J Pharmacol. 2002 Oct 25;453(2-3):209-15. PubMed PMID: 12398906.