TargetMol

PKC-theta inhibitor 1

Product Code:
 
TAR-T12496
Product Group:
 
Inhibitors and Activators
Supplier:
 
TargetMol
Regulatory Status:
 
RUO
Shipping:
 
cool pack
Storage:
 
-20℃
1 / 1
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CodeSizePrice
TAR-T12496-5mg5mg£703.00
Special offer! Add £1 to your order to get a TargetMol CCK-8 Kit. Read more here.
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TAR-T12496-50mg50mg£1,982.00
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Quantity:
TAR-T12496-100mg100mg£2,560.00
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This product comes from: United States.
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Further Information

Bioactivity:
PKC-theta inhibitor 1 is an inhibitor of PKC? (Ki of 6 nM)
CAS:
1160501-81-4
Formula:
C17H15F3N4O
Molecular Weight:
348.329
Pathway:
Chromatin/Epigenetic; Cytoskeletal Signaling
Purity:
0.98
SMILES:
NCC1(COC1)c1cccc(c1)-c1ccnc2[nH]nc(c12)C(F)(F)F
Target:
PKC

References

1. Collier PN, et al. Discovery of Selective, Orally Bioavailable Pyrazolopyridine Inhibitors of Protein Kinase C? (PKC?) That Ameliorate Symptoms of Experimental Autoimmune Encephalomyelitis. ACS Med Chem Lett. 2019 Jun 27;10(8):1134-1139.