PSB-12062

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TargetMol
Product Code: TAR-T12568
Supplier: TargetMol
CodeSizePrice
TAR-T12568-5mg5mg£108.00
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Quantity:
TAR-T12568-1mL1 mL * 10 mM (in DMSO)£112.00
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Quantity:
TAR-T12568-10mg10mg£128.00
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Quantity:
TAR-T12568-25mg25mg£201.00
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Quantity:
TAR-T12568-50mg50mg£293.00
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Quantity:
TAR-T12568-100mg100mg£462.00
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Quantity:
TAR-T12568-500mg500mg£922.00
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Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

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Documents

Further Information

Bioactivity:
PSB-12062 is a potent and selective antagonist of P2X4(IC50 of 1.38 μM for human P2X4).
CAS:
55476-47-6
Formula:
C19H15NO3S
Molecular Weight:
337.39
Pathway:
Membrane transporter/Ion channel; Neuroscience
Purity:
0.9997
SMILES:
Cc1ccc(cc1)S(=O)(=O)N1c2ccccc2Oc2ccccc12
Target:
P2X Receptor

References

1. Hernandez-Olmos V, et al. N-substituted phenoxazine and acridone derivatives: structure-activity relationships of potent P2X4 receptor antagonists. J Med Chem. 2012 Nov 26;55(22):9576-88. 2. Stokes L, et al. P2X4 Receptor Function in the Nervous System and Current Breakthroughs in Pharmacology.Front Pharmacol. 2017 May 23;8:291.