R-10015

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TargetMol
Product Code: TAR-T12609
Supplier: TargetMol
CodeSizePrice
TAR-T12609-1mg1mg£165.00
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TAR-T12609-2mg2mg£209.00
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TAR-T12609-5mg5mg£302.00
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TAR-T12609-1mL1 mL * 10 mM (in DMSO)£338.00
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TAR-T12609-10mg10mg£432.00
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TAR-T12609-25mg25mg£666.00
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TAR-T12609-50mg50mg£863.00
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TAR-T12609-100mg100mg£1,187.00
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TAR-T12609-500mg500mg£2,336.00
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Quantity:
Prices exclude any Taxes / VAT

Overview

Regulatory Status: RUO
Shipping:
cool pack
Storage:
-20℃

Images

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Documents

Further Information

Bioactivity:
R-10015 is a potent and selective inhibitor of LIM domain kinase (LIMK) and binds to the ATP-binding pocket(IC50 of 38 nM for human LIMK1),and a broad-spectrum antiviral compound for HIV infection.
CAS:
2097938-51-5
Formula:
C20H19ClN6O2
Molecular Weight:
410.86
Pathway:
Cell Cycle/Checkpoint; Microbiology/Virology
Purity:
0.9897
SMILES:
COC(=O)c1ccc2[nH]c(nc2c1)C1CCN(CC1)c1ncnc2[nH]cc(Cl)c12
Target:
LIM Kinase; Reverse Transcriptase

References

1. Yi F, et al. Discovery of Novel Small-Molecule Inhibitors of LIM Domain Kinase for Inhibiting HIV-1. J Virol. 2017 Jun 9;91(13). pii: e02418-16.